Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetRecQ-like DNA helicase BLM(Homo sapiens (Human))
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50440527(CHEMBL2426164)
Affinity DataIC50:  110nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional 3'-5' exonuclease/ATP-dependent helicase WRN(Homo sapiens (Human))
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50440527(CHEMBL2426164)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of WRN (unknown origin) by gel-based DNA unwinding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent DNA helicase Q1(Homo sapiens (Human))
National Center For Advancing Translational Sciences

Curated by ChEMBL
LigandPNGBDBM50440527(CHEMBL2426164)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of RECQ1 (unknown origin) by gel-based DNA unwinding assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed