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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
Boehringer Ingelheim International
US Patent
Ligand
BDBM158171
(US9029360, 14)
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Affinity Data
IC50: 603nM
Assay Description:
Activation of the mGluR5 receptor expressed in cell lines results in an increase in intracellular calcium concentration. Using calcium sensitive fluo...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
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US Patent
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Target
11-beta-hydroxysteroid dehydrogenase 1
(Homo sapiens (Human))
Boehringer Ingelheim International
US Patent
Ligand
BDBM158171
(US9029360, 14)
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Affinity Data
IC50: >1.00E+4nM
pH: 6.0 T: 2°C
Assay Description:
In vitro inhibition of 11beta -HSD1 was determined with HTRF (Homogeneous Time-Resolved Fluorescence) technology (cisbio international, France) detec...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI