Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384295(CHEMBL2030625)
Affinity DataKi:  22nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384295(CHEMBL2030625)
Affinity DataKi:  2.67E+3nMAssay Description:Inhibition of M5 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384295(CHEMBL2030625)
Affinity DataKi:  4.74E+3nMAssay Description:Inhibition of M2 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384295(CHEMBL2030625)
Affinity DataKi:  5.54E+3nMAssay Description:Inhibition of M1 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384295(CHEMBL2030625)
Affinity DataKi:  6.17E+3nMAssay Description:Inhibition of M4 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed