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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171936((2R,6S)-2,6-Bis-(2-naphthalen-1-yl-ethyl)-piperidi...)
Affinity DataKi:  4.68E+3nMAssay Description:Inhibition of 5 nM [3H]DTBZ binding to Vesicular Monoamine Transporter (VAMT2) of rat vesicle membranes More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50171936((2R,6S)-2,6-Bis-(2-naphthalen-1-yl-ethyl)-piperidi...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 3 nM [3H]-MLA binding to Nicotinic acetylcholine receptor alpha7 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed