Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 21 hits in this display
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
Ki: >1.00E+5nMAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
Ki: >1.00E+5nM ΔG°: >-23.7kJ/molepH: 7.5 T: 2°CAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
Ki: >1.00E+5nMAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: 22nMpH: 7.4 T: 2°CAssay Description:The compounds of the invention can be tested for their ability to inhibit LSD1. The ability of the compounds of the invention to inhibit LSD1 can be ...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: 22nMAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: 22nMAssay Description:The compounds of the invention can be tested for their ability to inhibit LSD1. The ability of the compounds of the invention to inhibit LSD1 can be ...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: 3.54E+4nMAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: 3.54E+4nMpH: 7.5 T: 2°CAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: 3.54E+4nMAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: >1.00E+5nMAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: >1.00E+5nMAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair
BDBM50142189(CHEMBL3759239 | US10329256, Example 5 | US9487512,...)
IC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:Human recombinant monoamine oxidase proteins MAO-A and MAO-B were purchased from Sigma Aldrich. MAOs catalyze the oxidative deamination of primary, s...More data for this Ligand-Target Pair