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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  7nMAssay Description:Displacement of [3H](+)-pentazocine from sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  661nMAssay Description:Inhibition of M3 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  696nMAssay Description:Inhibition of M2 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  802nMAssay Description:Inhibition of M5 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of M4 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  4.24E+3nMAssay Description:Inhibition of alpha2B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  4.26E+3nMAssay Description:Inhibition of alpha2C adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi:  7.96E+3nMAssay Description:Inhibition of M1 muscarinic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of alpha1B adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
The University Of Sydney

Curated by ChEMBL
LigandPNGBDBM50384286(CHEMBL2030626)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of D3 dopamine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed