Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 5(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111159(3-Piperazin-1-ylmethyl-1H-indole | CHEMBL276397)
Affinity DataKi:  2.56E+5nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 5 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111159(3-Piperazin-1-ylmethyl-1H-indole | CHEMBL276397)
Affinity DataKi: >1.00E+6nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 4 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111159(3-Piperazin-1-ylmethyl-1H-indole | CHEMBL276397)
Affinity DataKi: >1.00E+6nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 1 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50111159(3-Piperazin-1-ylmethyl-1H-indole | CHEMBL276397)
Affinity DataKi: >1.00E+6nMAssay Description:Tested for its binding affinity towards human recombinant Melanocortin 3 receptor by using radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed