Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50137532(CHEMBL3752965)
Affinity DataKi:  375nMAssay Description:Displacement of [3H]HEMADO from human A3 adenosine receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50137532(CHEMBL3752965)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]NECA from human A2A adenosine receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50137532(CHEMBL3752965)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]CCPA from human A1 adenosine receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50137532(CHEMBL3752965)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity at human A2B adenosine receptor expressed in CHO cell membranes assessed as inhibition of NECA stimulated adenylyl cyclase activi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed