Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170943(Benzyl-(2-phenyl-2H-pyrazolo[4,3-c]quinolin-4-yl)-...)
Affinity DataKi:  125nMAssay Description:Inhibition of [3H]-MRE3008-F20 binding to human adenosine A3 receptor expressed in CHO cells; (n=3 - 6)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170943(Benzyl-(2-phenyl-2H-pyrazolo[4,3-c]quinolin-4-yl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-ZM-241,385 binding to human adenosine A2a receptor expressed in CHO cells; (n=3 - 6)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170943(Benzyl-(2-phenyl-2H-pyrazolo[4,3-c]quinolin-4-yl)-...)
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of [3H]-DPCPX binding to human adenosine A1 receptor expressed in CHO cells; (n=3 - 6)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50170943(Benzyl-(2-phenyl-2H-pyrazolo[4,3-c]quinolin-4-yl)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of 100 nM-NECA stimulation of cAMP levels in human adenosine A2b receptor expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed