Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50328010(3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridi...)
Affinity DataIC50:  470nMAssay Description:Inactivation of nAChR alpha4beta2 in human SH-EP1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University Of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50328010(3-[(2(S)-Azetidinyl)methoxy]-5-(piperidinyl)pyridi...)
Affinity DataEC50:  1.14E+3nMAssay Description:Agonist activity at human nAChR alpha4beta2 in human SH-EP1 cells assessed as induction in rubidium effluxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed