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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5
(RAT)
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50366538
(CHEMBL1169506)
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Affinity Data
IC50: 41nM
Assay Description:
Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligand
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50366538
(CHEMBL1169506)
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Copy InChI
Affinity Data
EC50: 159nM
Assay Description:
Stimulation of phosphoinositide hydrolysis in A9L cells expressing human m1 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50366538
(CHEMBL1169506)
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Copy InChI
Affinity Data
EC50: 1.08E+3nM
Assay Description:
Stimulation of cAMP in CHO cells expressing human m2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI