Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM50301288(2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepi...)
BDBM50301288(2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepi...)
Ki: 2.70E+3nMAssay Description:Displacement of [3H]-mesulergine from recombinant human 5-HT2C receptor transfected in Swiss mouse 3T3 cells after 150 mins by scintillation proximit...More data for this Ligand-Target Pair
BDBM50301288(2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepi...)
EC50: 4.98E+3nMAssay Description:Agonist activity at recombinant human 5-HT2C receptor transfected in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
BDBM50301288(2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepi...)
EC50: 4.98E+3nMAssay Description:Agonist activity at recombinant human 5-HT2C receptor transfected in CHOK1 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
BDBM50301288(2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepi...)
EC50: 4.98E+3nMAssay Description:Agonist activity at human recombinant 5HT2C receptor expressed in CHO K1 cells assessed as induction of calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
BDBM50301288(2-benzyl-2,4,5,6,7,8-hexahydropyrazolo[4,3-d]azepi...)