Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetTyrosine-protein kinase ITK/TSK [357-620,Y512E](Homo sapiens (Human))
Glaxosmithkline

LigandBDBM213224(N2-[(3R)-1-Acryloyl-3-pyrrolidinyl]-6-(4-morpholin...)Copy SMILESCopy InChI

Affinity DataIC50:  2.00E+4nMAssay Description:This assay is based on the binding and displacement of Alexa-fluor 647-labeled ATP-competitive kinase inhibitor tracer 236. Binding of the tracer is ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI