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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50058045(CHEMBL3330813)
Affinity DataIC50:  128nMAssay Description:Antagonist activity at mGluR1 (unknown origin) expressed in Chem-3 cells assessed as inhibition of glutamate-induced increased intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed