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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  100nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medulla using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(BOVINE)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from bovine kidney inner medullaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a/V1b receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed