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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSigma non-opioid intracellular receptor 1(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50080950((R)-2-(4-(3-fluorobenzyloxy)benzylamino)propanamid...)
Affinity DataIC50:  280nMAssay Description:Inhibition of [3H]pentazocine binding to Opioid receptor sigma 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50080950((R)-2-(4-(3-fluorobenzyloxy)benzylamino)propanamid...)
Affinity DataIC50:  450nMAssay Description:Inhibition of rat brain mitochondria MAOB by radioenzymatic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50080950((R)-2-(4-(3-fluorobenzyloxy)benzylamino)propanamid...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of [3H]batrachotoxin binding to rat brain sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University Of Bari

Curated by ChEMBL
LigandPNGBDBM50080950((R)-2-(4-(3-fluorobenzyloxy)benzylamino)propanamid...)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of rat brain mitochondria MAOA by radioenzymatic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50080950((R)-2-(4-(3-fluorobenzyloxy)benzylamino)propanamid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of [3H]saxitoxin binding to rat brain sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed