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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
17-beta-hydroxysteroid dehydrogenase type 3
(Homo sapiens (Human))
Chuq (Chul)-Research Center
Curated by
ChEMBL
Ligand
BDBM50350421
(CHEMBL1813731)
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Affinity Data
IC50: 6nM
Assay Description:
Inhibition of 17Beta-HSD3 expressed in intact HEK293 cells assessed as transformation of [14C]-4-androstene-3,17-dione into [14C]-testosterone in pre...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
17-beta-hydroxysteroid dehydrogenase type 3
(Homo sapiens (Human))
Chuq (Chul)-Research Center
Curated by
ChEMBL
Ligand
BDBM50350421
(CHEMBL1813731)
Copy SMILES
Copy InChI
Affinity Data
IC50: 6nM
Assay Description:
Inhibition of 17betaHSD3 (unknown origin) transfected in HEK293 cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
17-beta-hydroxysteroid dehydrogenase type 3
(Rattus norvegicus)
Chu De Qu£Bec-Research Center (Chul)
Curated by
ChEMBL
Ligand
BDBM50350421
(CHEMBL1813731)
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Copy InChI
Affinity Data
IC50: 13nM
Assay Description:
Inhibition of 17beta-HSD3 in rat testes microsomes using [14C]-4-androstene-3,17-dione as substrate after 2 hrs
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
17-beta-hydroxysteroid dehydrogenase type 3
(Homo sapiens (Human))
Chuq (Chul)-Research Center
Curated by
ChEMBL
Ligand
BDBM50350421
(CHEMBL1813731)
Copy SMILES
Copy InChI
Affinity Data
IC50: 85nM
Assay Description:
Inhibition of 17betaHSD3 (unknown origin) transfected in human LNCAP cells assessed as conversion of [14C]-4-androstene-3,17-dione into [14C]-testost...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
17-beta-hydroxysteroid dehydrogenase type 3
(Homo sapiens (Human))
Chuq (Chul)-Research Center
Curated by
ChEMBL
Ligand
BDBM50350421
(CHEMBL1813731)
Copy SMILES
Copy InChI
Affinity Data
IC50: 110nM
Assay Description:
Inhibition of 17-beta-HSD3 (unknown origin) expressed in human LNCaP cells using [14C]-4-androstene-3,17-dione as substrate assessed as reduction of ...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI