Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50042462(1-(4-Dimethylamino-but-2-ynyl)-4-methyl-pyrrolidin...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50042462(1-(4-Dimethylamino-but-2-ynyl)-4-methyl-pyrrolidin...)
Affinity DataKi:  1.50E+4nMAssay Description:Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50042462(1-(4-Dimethylamino-but-2-ynyl)-4-methyl-pyrrolidin...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50042462(1-(4-Dimethylamino-but-2-ynyl)-4-methyl-pyrrolidin...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50042462(1-(4-Dimethylamino-but-2-ynyl)-4-methyl-pyrrolidin...)
Affinity DataKi:  1.50E+5nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed