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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
7Tm Pharma
Curated by
ChEMBL
Ligand
BDBM50177296
((R)-N-(4-methyl-2-(3-methylpiperazin-1-yl)quinolin...)
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Affinity Data
IC50: 4.10nM
Assay Description:
Displacement of [125I]MCH from human MCH1 receptor expressed in CHO cell by WC assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
7Tm Pharma
Curated by
ChEMBL
Ligand
BDBM50177296
((R)-N-(4-methyl-2-(3-methylpiperazin-1-yl)quinolin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 18nM
Assay Description:
Inhibition of human MCH1 receptor by SPA assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanin-concentrating hormone receptor 1
(Homo sapiens (Human))
7Tm Pharma
Curated by
ChEMBL
Ligand
BDBM50177296
((R)-N-(4-methyl-2-(3-methylpiperazin-1-yl)quinolin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Displacement of [3H]myo-inositol from human MCH1 receptor expressed in CHO cell by IP3 assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI