Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 20 hits in this display
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
IC50: 0.372nMAssay Description:Compounds were screened for their ability to displace a fluorescent labelled tracer ERβ ligand via time resolved fluorescent energy transfer usi...More data for this Ligand-Target Pair
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
IC50: <0.640nMAssay Description:Compounds were screened for their ability to displace a fluorescent labelled tracer ERβ ligand via time resolved fluorescent energy transfer usi...More data for this Ligand-Target Pair
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
IC50: 1nMAssay Description:Compounds were screened for their ability to displace a fluorescent labelled tracer ERβ ligand via time resolved fluorescent energy transfer usi...More data for this Ligand-Target Pair
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)
BDBM50125052(CHEMBL3623004 | US10130617, Example 1 | WO-2014/19...)