Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataEC50:  1.09E+4nMAssay Description:Effective concentration against mouse melanocortin MC4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataEC50:  2.22E+3nMAssay Description:Effective concentration against mouse Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50144870(CHEMBL410091 | Tyr-c[Asp-Trp-Arg-DPhe-Asn-Ala-Phe-...)
Affinity DataEC50:  6.12E+3nMAssay Description:Effective concentration against mouse Melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed