Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM50339346((R)-trans-(2S,5S,8S,11S,14R,19R,22S,25R,28R,31S)-2...)
EC50: 85nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
BDBM50339346((R)-trans-(2S,5S,8S,11S,14R,19R,22S,25R,28R,31S)-2...)
EC50: 495nMAssay Description:Agonist activity at mouse melanocortin 3 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
BDBM50339346((R)-trans-(2S,5S,8S,11S,14R,19R,22S,25R,28R,31S)-2...)
EC50: 72nMAssay Description:Agonist activity at mouse melanocortin 5 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
BDBM50339346((R)-trans-(2S,5S,8S,11S,14R,19R,22S,25R,28R,31S)-2...)
EC50: 33nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair