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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetN-acylethanolamine-hydrolyzing acid amidase(Rattus norvegicus (Rat))
University Of California

US Patent
LigandPNGBDBM50032460(CHEMBL3353550 | US9353075, 3)
Affinity DataIC50:  1.21E+3nMpH: 7.4Assay Description:Lysosomal NAAA protein preparation were obtained by homogenizing male Sprague-Dawley rat lungs (Charles River) in 20 mM Tris-HCl buffer pH 7.4 contai...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetN-acylethanolamine-hydrolyzing acid amidase(Rattus norvegicus (Rat))
University Of California

US Patent
LigandPNGBDBM50032460(CHEMBL3353550 | US9353075, 3)
Affinity DataIC50:  1.22E+3nMAssay Description:Inhibition of NAAA in Sprague-Dawley rat lung assessed as inhibition of hydrolysis of 10-cis-heptadecenoylethanolamide by UPLC/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acylethanolamine-hydrolyzing acid amidase(Rattus norvegicus (Rat))
University Of California

US Patent
LigandPNGBDBM50032460(CHEMBL3353550 | US9353075, 3)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of NAAA in Sprague-Dawley rat lung assessed as inhibition of hydrolysis of 10-cis-heptadecenoylethanolamide by UPLC/MS methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed