Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAndrogen receptor(Homo sapiens (Human))
Bayer Intellectual Property Gbmh

US Patent

LigandBDBM150276(US8987239, 1)Copy SMILESCopy InChI

Affinity DataIC50:  6nMAssay Description:The test was carried out as in 1, with the following modifications: cytosol from androgen receptor-expressing insect cells (Hi5) was used, and the re...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails US Patent
Copy BDB DOI

TargetProgesterone receptor(Homo sapiens (Human))
Bayer Intellectual Property Gbmh

US Patent

LigandBDBM150276(US8987239, 1)Copy SMILESCopy InChI

Affinity DataIC50:  15nMAssay Description:Using cytosol from progesterone receptor-expressing insect cells (Hi5), competitive binding to the progesterone receptor was determined from the abil...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails US Patent
Copy BDB DOI