Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50205508((R,R)-(+)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydro...)
Affinity DataKi:  501nMAssay Description:Displacement of [125I]CYP from human adrenergic beta 2 receptor transfected in CHO cells in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50205508((R,R)-(+)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydro...)
Affinity DataKi:  6.46E+3nMAssay Description:Displacement of [125I]CYP from human adrenergic beta 1 receptor transfected in CHO cells in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50205508((R,R)-(+)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydro...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [125I]CYP from human adrenergic beta 3 receptor transfected in CHO cells in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed