Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123442((4-Methyl-4-{(S)-3-methyl-4-[(S)-1-(4-trifluoromet...)
Affinity DataKi:  10nMAssay Description:Ability to inhibit [125I]-labeled RANTES binding to the CCR5 receptor expressed in membrane preparations from CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123442((4-Methyl-4-{(S)-3-methyl-4-[(S)-1-(4-trifluoromet...)
Affinity DataKi:  10nMAssay Description:Inhibition of RANTES binding to the human C-C chemokine receptor type 5 (CCR5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50123442((4-Methyl-4-{(S)-3-methyl-4-[(S)-1-(4-trifluoromet...)
Affinity DataKi:  985nMAssay Description:Binding affinity towards muscarinic receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed