Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 18 hits in this display   

TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  3.70E+4nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  2.20E+5nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytosol aminopeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition against Leucyl aminopeptidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  1.70E+6nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition against cytosolic Aminopeptidase P from human heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >3.00E+6nMAssay Description:Inhibition against cytosolic Aminopeptidase P from human heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 1(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition against cytosolic Aminopeptidase P from human heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition against membrane bound monkey aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Inhibition against membrane bound human aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro aminopeptidase 2(Rattus norvegicus)
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+6nMAssay Description:Activity against membrane bound rat aminopeptidase PMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+7nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
Pharmacia And Upjohn

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+7nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed