Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetClan CD, family C13, asparaginyl endopeptidase-like cysteine peptidase(Trichomonas vaginalis G3)
Georgia Institute Of Technology

LigandPNGBDBM22126(aza-peptide Michael acceptor, 5j | benzyl N-[(1S)-...)
Affinity DataIC50: <1nMT: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Ixodes ricinus)
Georgia Institute Of Technology

LigandPNGBDBM22126(aza-peptide Michael acceptor, 5j | benzyl N-[(1S)-...)
Affinity DataIC50:  5.5nMT: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLegumain(Schistosoma mansoni)
Georgia Institute Of Technology

LigandPNGBDBM22126(aza-peptide Michael acceptor, 5j | benzyl N-[(1S)-...)
Affinity DataIC50:  35nMpH: 6.8 T: 2°CAssay Description:AE activity in the induction medium was measured with the substrate Cbz-Ala-Ala-Asn-AMC. In a black 96-well microtiter plate, aza-peptidyl inhibitors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed