Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A1(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg

Curated by ChEMBL
LigandPNGBDBM50051661(2-(3,4-Dichloro-phenyl)-5,6-dimethyl-7-((R)-1-phen...)
Affinity DataKi:  330nMAssay Description:Radioligand binding assay for [3H]-PIA affinity towards Adenosine A1 receptor of rat cerebral cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Julius-Maximilians-UniversitäT WüRzburg

Curated by ChEMBL
LigandPNGBDBM50051661(2-(3,4-Dichloro-phenyl)-5,6-dimethyl-7-((R)-1-phen...)
Affinity DataKi: >3.00E+4nMAssay Description:Radioligand binding assay for [3H]-NECA affinity towards adenosine A2A receptor of rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed