Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 9 hits in this display
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
Ki: 1.5nMAssay Description:Binding affinity was determined against Opioid receptor mu 1 obtained from guinea pig brain membranes using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
Ki: 1.5nMAssay Description:Binding affinity was determined against Opioid receptor mu 1 obtained from guinea pig brain membranes using [3H]DAMGO as radioligandMore data for this Ligand-Target Pair
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
Ki: 4.70nMAssay Description:Binding affinity was determined against Opioid receptor kappa 1 obtained from guinea pig brain membranes using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
Ki: 4.70nMAssay Description:Binding affinity was determined against Opioid receptor kappa 1 obtained from guinea pig brain membranes using [3H]U-69593 as radioligandMore data for this Ligand-Target Pair
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
Ki: 54nMAssay Description:Binding affinity was determined against Opioid receptor delta 1 obtained from guinea pig brain membranes using [3H]naltrindole as radioligandMore data for this Ligand-Target Pair
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
BDBM50085021(Benzyl-((6S,11R)-3-cyclopropylmethyl-6,11-dimethyl...)
Ki: 57nMAssay Description:Binding affinity was determined against Opioid receptor delta 1 obtained from guinea pig brain membranes using [3H]naltrindole as radioligandMore data for this Ligand-Target Pair