Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50315668(((3R,4S)-4-(2,4-difluorophenyl)-1-(pyrimidin-2-yl)...)
BDBM50315668(((3R,4S)-4-(2,4-difluorophenyl)-1-(pyrimidin-2-yl)...)
EC50: 243nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in CHO cells by cAMP responsive beta lactamase reporter gene assayMore data for this Ligand-Target Pair
BDBM50315668(((3R,4S)-4-(2,4-difluorophenyl)-1-(pyrimidin-2-yl)...)
EC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant MC1 receptor expressed in HEK293 cells assessed as cAMP accumulation by enzyme fragment complementation assayMore data for this Ligand-Target Pair
BDBM50315668(((3R,4S)-4-(2,4-difluorophenyl)-1-(pyrimidin-2-yl)...)
EC50: >2.67E+4nMAssay Description:Agonist activity at human recombinant MC3 receptor expressed in CHO cells assessed as cAMP accumulation by enzyme fragment complementation assayMore data for this Ligand-Target Pair
BDBM50315668(((3R,4S)-4-(2,4-difluorophenyl)-1-(pyrimidin-2-yl)...)
EC50: >1.11E+4nMAssay Description:Agonist activity at human recombinant MC5 receptor expressed in HEK293 cells assessed as cAMP accumulation by beta lactamase reporter gene assayMore data for this Ligand-Target Pair