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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
Research Triangle Institute
Curated by
ChEMBL
Ligand
BDBM50064526
(3-((3R,4R)-1-Cyclopentyl-3,4-dimethyl-piperidin-4-...)
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Affinity Data
Ki: 199nM
Assay Description:
Inhibition of [3H]U69,593 binding to Opioid receptor kappa 1 of guinea pig membranes
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Research Triangle Institute
Curated by
ChEMBL
Ligand
BDBM50064526
(3-((3R,4R)-1-Cyclopentyl-3,4-dimethyl-piperidin-4-...)
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Affinity Data
Ki: 444nM
Assay Description:
Inhibition of [3H]-DAMGO binding to Opioid receptor mu 1 of rat brain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Research Triangle Institute
Curated by
ChEMBL
Ligand
BDBM50064526
(3-((3R,4R)-1-Cyclopentyl-3,4-dimethyl-piperidin-4-...)
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Copy InChI
Affinity Data
Ki: >7.30E+3nM
Assay Description:
Inhibition of [3H]-DADLE binding to Opioid receptor delta 1 of rat brain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI