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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Muscarinic acetylcholine receptor M1
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50223980
(3-(benzyl-phenyl-carbamoyloxy)-8,8-dimethyl-8-azon...)
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Affinity Data
IC50: 4.5nM
Assay Description:
Antagonist activity at cloned muscarinic M1 receptor expressed in CHO cells by measuring calcium mobilization
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M3
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50223980
(3-(benzyl-phenyl-carbamoyloxy)-8,8-dimethyl-8-azon...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.60nM
Assay Description:
Antagonist activity at cloned muscarinic M3 receptor expressed in CHO cells by measuring calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(Homo sapiens (Human))
Glaxosmithkline
Curated by
ChEMBL
Ligand
BDBM50223980
(3-(benzyl-phenyl-carbamoyloxy)-8,8-dimethyl-8-azon...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 48nM
Assay Description:
Antagonist activity at cloned muscarinic M2 receptor expressed in CHO cells by measuring calcium mobilization
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI