Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 17 hits in this display
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
IC50: 3.20E+4nMAssay Description:Inhibition of Cdc42 GTPase activity assessed as incorporation of BODIPY-GTP after 40 mins by nucleotide binding competition assayMore data for this Ligand-Target Pair
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
IC50: 5.80E+4nMAssay Description:Inhibition of Rac1 GTPase activity assessed as incorporation of BODIPY-GTP after 40 mins by nucleotide binding competition assayMore data for this Ligand-Target Pair
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
IC50: >1.00E+5nMAssay Description:Inhibition of RGS17 (unknown origin) C117A mutant interaction with biotinylated Galphao after 30 mins in presence of AMF and GDP by AlphaScreen assayMore data for this Ligand-Target Pair
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
IC50: 2.00E+5nMAssay Description:Inhibition of recombinant human DOPA decarboxylase assessed as inhibition of dopamine production after 30 mins by HPLC methodMore data for this Ligand-Target Pair
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)
BDBM25525(24-methyl-5,7,18,20-tetraoxa-24-azahexacyclo[11.11...)