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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
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Target
Lysine-specific histone demethylase 1A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
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Affinity Data
IC50: 11nM
pH: 7.5 T: 2°C
Assay Description:
The LSD1 screening biochemical assay was performed by Shanghai ChemPartner Co. Ltd and the detailed protocol was shown as followed. The AlphaLISA ass...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
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MCE
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Lysine-specific histone demethylase 1A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 13nM
Assay Description:
The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific histone demethylase 1A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 13nM
Assay Description:
The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Lysine-specific histone demethylase 1A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <50nM
Assay Description:
The purpose of this test is to test the in vitro inhibitory activities of the compounds against LSD1. The enzyme used in this experiment was human LS...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Utah Research Foundation
US Patent
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
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Affinity Data
IC50: >3.00E+5nM
Assay Description:
Inhibition of monoamine oxidase activity was carried used using the MAO-Glo.TM. Assay Kit according to the manufacturer's suggested protocol. Bri...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
University Of Utah Research Foundation
US Patent
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
Copy SMILES
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Affinity Data
IC50: >3.00E+5nM
Assay Description:
Inhibition of monoamine oxidase activity was carried used using the MAO-Glo.TM. Assay Kit according to the manufacturer's suggested protocol. Bri...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
University Of Utah Research Foundation
US Patent
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+5nM
Assay Description:
Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
University Of Utah Research Foundation
US Patent
Ligand
BDBM151611
(SP-2509 | US11433053, Example HCI-2509 | US8987335...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >3.00E+5nM
Assay Description:
Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
MCE
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI