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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target3-oxoacyl-[acyl-carrier-protein] synthase 1 [C171Q](Mycobacterium tuberculosis)
University Of Wuerzburg

LigandPNGBDBM214777(TLM18)
Affinity DataKi:  3.84E+5nMpH: 8.5Assay Description:Binding of TLM18 to wild-type and mutant KasA was quantified by monitoring changes in the intrinsic tryptophan fluorescence of the enzyme at waveleng...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
Target3-oxoacyl-[acyl-carrier-protein] synthase 2(Staphylococcus aureus)
Colorado State University

Curated by ChEMBL
LigandPNGBDBM214777(TLM18)
Affinity DataKd:  1.07E+5nMAssay Description:Binding affinity to Staphylococcus aureus wild type FabF expressed in Escherichia coli BL21 (DE3) PlysS cells by intrinsic tryptophan fluorescence qu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 2(Staphylococcus aureus)
Colorado State University

Curated by ChEMBL
LigandPNGBDBM214777(TLM18)
Affinity DataKd:  1.07E+5nMAssay Description:Binding affinity to Staphylococcus aureus wild type FabF expressed in Escherichia coli BL21 (DE3) PlysS cells by intrinsic tryptophan fluorescence qu...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
Target3-oxoacyl-[acyl-carrier-protein] synthase 1(Mycobacterium tuberculosis)
University Of Wuerzburg

LigandPNGBDBM214777(TLM18)
Affinity DataKd:  1.12E+5nMpH: 8.5Assay Description:Binding of TLM18 to wild-type and mutant KasA was quantified by monitoring changes in the intrinsic tryptophan fluorescence of the enzyme at waveleng...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB