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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  35nMAssay Description:Compound was tested for inhibitory activity against ACAT from canine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  36nMAssay Description:Compound was tested for inhibitory activity against ACAT from rabbit liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  36nMAssay Description:Compound was tested for inhibitory activity against ACAT from canine adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  43nMAssay Description:Compound was tested for inhibitory activity against ACAT from rabbit liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  45nMAssay Description:Compound was tested for inhibitory activity against ACAT from rabbit intestineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  56nMAssay Description:Compound was tested for inhibitory activity against ACAT from canine intestineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  228nMAssay Description:Compound was tested for inhibitory activity against ACAT from Caco-2 microsome in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  3.57E+3nMAssay Description:Compound was tested for inhibitory activity against ACAT from canine liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSterol O-acyltransferase 1(Homo sapiens (Human))
Azwell

Curated by ChEMBL
LigandPNGBDBM50079716((5E,8E,11E,14E,17E,20E)-Docosa-5,8,11,14,17,20-hex...)
Affinity DataIC50:  7.24E+3nMAssay Description:Compound was tested for inhibitory activity against ACAT from U937 microsome in humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed