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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86831((+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86831((+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86831((+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  251nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed