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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Adenosine receptor A1
(BOVINE)
Center For Bio-Pharmaceutical Sciences
Curated by
ChEMBL
Ligand
BDBM50011596
((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
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Affinity Data
Ki: 23nM
Assay Description:
Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Adenosine receptor A1
(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences
Curated by
ChEMBL
Ligand
BDBM50011596
((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
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Copy InChI
Affinity Data
Ki: 230nM
Assay Description:
Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A3
(Homo sapiens (Human))
Leiden University
Curated by
ChEMBL
Ligand
BDBM50011596
((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
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Affinity Data
Ki: 786nM
Assay Description:
Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membrane
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Adenosine receptor A2a
(Homo sapiens (Human))
Leiden University
Curated by
ChEMBL
Ligand
BDBM50011596
((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
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Affinity Data
Ki: 3.15E+3nM
Assay Description:
Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A1
(Homo sapiens (Human))
Leiden University
Curated by
ChEMBL
Ligand
BDBM50011596
((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.42E+3nM
Assay Description:
Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI