Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAdenosine receptor A1(BOVINE)
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of calf brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Center For Bio-Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]CPX from adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  786nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  3.15E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50011596((2-Cyclopentyl-1H-imidazo[4,5-c]quinolin-4-yl)-phe...)
Affinity DataKi:  3.42E+3nMAssay Description:Displacement of [3H]R-PIA from human adenosine A1 receptor in CHO membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed