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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  41nMAssay Description:Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  64nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cellsMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  219nMAssay Description:Binding affinity for human Alpha-2B adrenergic receptor from cultured Y-1 cells using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  309nMAssay Description:Binding affinity for human Alpha-2A adrenergic receptor from cultured LM(tk-) cells using [3H]rauwolscineMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  1.41E+3nMAssay Description:Binding affinity for human Alpha-2C adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  3.24E+3nMAssay Description:Binding affinity for human Alpha-1B adrenergic receptor from cultured LM(tk-) cells using [3H]prazosin More data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in human brainMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity for Alpha-1 adrenergic receptor of human cerebral cortex membraneMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  1.23E+4nMAssay Description:Binding affinity for human Alpha-1D adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosinMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50213029(CHEMBL49395)
Affinity DataKi:  1.82E+4nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor from cultured LM(tk-) cells using [3H]-prazosinMore data for this Ligand-Target Pair
In DepthDetails