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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
10
hits in this display
Target
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
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Affinity Data
Ki: 41nM
Assay Description:
Binding affinity for Alpha-2 adrenergic receptor of CHO-C10 membrane preparation
More data for this Ligand-Target Pair
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Target
Alpha-2A/Alpha-2B/Alpha-2C adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 64nM
Assay Description:
Binding affinity towards Alpha-2 adrenergic receptor in HT-29 cells
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-2B adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
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Affinity Data
Ki: 219nM
Assay Description:
Binding affinity for human Alpha-2B adrenergic receptor from cultured Y-1 cells using [3H]rauwolscine
More data for this Ligand-Target Pair
Target Info
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Target
Alpha-2A adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 309nM
Assay Description:
Binding affinity for human Alpha-2A adrenergic receptor from cultured LM(tk-) cells using [3H]rauwolscine
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
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Copy BDB DOI
Target
Alpha-2C adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.41E+3nM
Assay Description:
Binding affinity for human Alpha-2C adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosin
More data for this Ligand-Target Pair
Target Info
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Reactome pathway
UniProtKB/SwissProt
antibodypedia
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Copy BDB DOI
Target
Alpha-1B adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.24E+3nM
Assay Description:
Binding affinity for human Alpha-1B adrenergic receptor from cultured LM(tk-) cells using [3H]prazosin
More data for this Ligand-Target Pair
Target Info
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
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Copy BDB DOI
Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
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Copy InChI
Affinity Data
Ki: 1.10E+4nM
Assay Description:
Binding affinity towards Alpha-1 adrenergic receptor in human brain
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
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antibodypedia
antibodypedia
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CHEMBL
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In Depth
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Copy BDB DOI
Target
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.10E+4nM
Assay Description:
Binding affinity for Alpha-1 adrenergic receptor of human cerebral cortex membrane
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
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antibodypedia
antibodypedia
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In Depth
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Copy BDB DOI
Target
Alpha-1D adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.23E+4nM
Assay Description:
Binding affinity for human Alpha-1D adrenergic receptor from cultured LM(tk-) cells using [3H]- prazosin
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
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DrugBank
antibodypedia
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CHEMBL
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In Depth
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Copy BDB DOI
Target
Alpha-1A adrenergic receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM50213029
(CHEMBL49395)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.82E+4nM
Assay Description:
Binding affinity for human Alpha-1A adrenergic receptor from cultured LM(tk-) cells using [3H]-prazosin
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Copy BDB DOI