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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Targacept
Curated by
ChEMBL
Ligand
BDBM50309862
(4-Benzoxazo-2-yl-1,4-diazabicyclo[3.2.2]nonane | C...)
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Affinity Data
Ki: 13nM
Assay Description:
Binding affinity to 5HT3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 3A
(Mus musculus (house mouse))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50309862
(4-Benzoxazo-2-yl-1,4-diazabicyclo[3.2.2]nonane | C...)
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Copy InChI
Affinity Data
Ki: 13nM
Assay Description:
Displacement of [3H]LY278584 from mouse 5HT3 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuronal acetylcholine receptor subunit alpha-7
(Rattus norvegicus (Rat))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50309862
(4-Benzoxazo-2-yl-1,4-diazabicyclo[3.2.2]nonane | C...)
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Copy InChI
Affinity Data
Ki: 22.5nM
Assay Description:
Displacement of [125I]BTX from rat alpha7 nicotinic acetylcholine receptor expressed in GH4C1 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuronal acetylcholine receptor subunit alpha-7
(Homo sapiens (Human))
Targacept
Curated by
ChEMBL
Ligand
BDBM50309862
(4-Benzoxazo-2-yl-1,4-diazabicyclo[3.2.2]nonane | C...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 22.5nM
Assay Description:
Binding affinity to alpha7 nAChR
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI