Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156719(2-(1-benzoyl-4-piperidinyl)-2-{[4-(2-butynyloxy)ph...)
Affinity DataIC50:  233nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156719(2-(1-benzoyl-4-piperidinyl)-2-{[4-(2-butynyloxy)ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156719(2-(1-benzoyl-4-piperidinyl)-2-{[4-(2-butynyloxy)ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50156719(2-(1-benzoyl-4-piperidinyl)-2-{[4-(2-butynyloxy)ph...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed