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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  2nMAssay Description:Inhibition of TACEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  35nMAssay Description:Inhibition of MMP8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  96nMAssay Description:Inhibition of MMP13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-14(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  582nMAssay Description:Inhibition of MMP14More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  777nMAssay Description:Inhibition of MMP9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrilysin(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  961nMAssay Description:Inhibition of MMP7More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisintegrin and metalloproteinase domain-containing protein 10(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of ADAM10More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInterstitial collagenase(Homo sapiens (Human))
University Of Athens

Curated by ChEMBL
LigandPNGBDBM50264814((2R,3S)-2-(4-(but-2-ynyloxy)phenylsulfonamido)-N,3...)
Affinity DataIC50:  2.47E+3nMAssay Description:Inhibition of MMP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed