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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50165928
(Ac-[CEHdFRWC]-NH2 | CHEMBL385556)
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Affinity Data
Ki: 2.30nM
Assay Description:
Inhibition of [125I]-NDP-alpha-MSH binding to melanocortin-4 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50165928
(Ac-[CEHdFRWC]-NH2 | CHEMBL385556)
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Copy InChI
Affinity Data
Ki: 67nM
Assay Description:
Inhibition of [125I]NDP-alpha-MSH binding to melanocortin-1 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50165928
(Ac-[CEHdFRWC]-NH2 | CHEMBL385556)
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Copy InChI
Affinity Data
Ki: 400nM
Assay Description:
Inhibition of [125I]-NDP-alpha-MSH binding to melanocortin-3 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50165928
(Ac-[CEHdFRWC]-NH2 | CHEMBL385556)
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Copy InChI
Affinity Data
Ki: >500nM
Assay Description:
Inhibition of [125I]NDP-alpha-MSH binding to melanocortin-5 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50165928
(Ac-[CEHdFRWC]-NH2 | CHEMBL385556)
Copy SMILES
Copy InChI
Affinity Data
EC50: 0.300nM
Assay Description:
Agonist activity at human Melanocortin-4 receptor as peptide required for 50% maximal cAMP release (n > or =2)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI