Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Ki: 6nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Ki: 120nMpH: 7.5Assay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Ki: 120nM ΔG°: -41.1kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Ki: 120nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
BDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
EC50: 0.5nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair