Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  6nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  6nM ΔG°:  -48.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  6nMpH: 7.5Assay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  6nMAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  6nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  120nMpH: 7.5Assay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  120nM ΔG°:  -41.1kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataKi:  120nMAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataEC50:  18nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanocortin receptor 4(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM135767(US10179804, Example 152 | US10632171, Peptide No. ...)
Affinity DataEC50:  0.5nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In DepthDetails US Patent