Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50331211(1-(2-acetyl-5-methyl-2,3,4,5-tetrahydro-1H-pyrido[...)
Affinity DataKi:  168nMAssay Description:Displacement of [3H]4-(benzyloxy)-1-(1-(2-(pyrrolidin-1-yl)ethyl)-1H-indazol-5-yl)pyridin-2(1H)-one from MCH-1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed