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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50140506
((E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cy...)
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Affinity Data
IC50: 63nM
Assay Description:
Antagonist activity at NPYY2 receptor (unknown origin) assessed as inhibition of PYY-induced [33S]-GTPgammaS binding
More data for this Ligand-Target Pair
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Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50140506
((E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cy...)
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Copy InChI
Affinity Data
IC50: 63.1nM
Assay Description:
Antagonist activity at human neuropeptide Y2 receptor by [35]GTPgammaS assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50140506
((E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Displacement of [125I]-NPY from NPYY2 receptor (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50140506
((E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Binding affinity to neuropeptide Y2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50140506
((E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Binding affinity towards human NPY Y2 receptor was determined using [35S]-GTP-gammaS, radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Neuropeptide Y receptor type 2
(Homo sapiens (Human))
The Scripps Research Institute
Curated by
ChEMBL
Ligand
BDBM50140506
((E)-N-(1-Acetyl-2,3-dihydro-1H-indol-6-yl)-3-(3-cy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Displacement of [125I]PYY from human NPY Y2 receptor expressed endogenously in KAN-Ts cells by scintillation counting
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI