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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity for human Melatonin receptor type 1A stably transfected in human embryonic kidney cells (HEK 293) using 2-[125I]-iodomelatonin as ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  112nMAssay Description:Binding affinity to MT2 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  112nMAssay Description:Binding affinity for human Melatonin receptor type 1B stably transfected in human embryonic kidney cells (HEK 293) using 2-[125I]-iodomelatonin as ra...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  149nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed