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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50007171(CHEMBL316090 | N-(4-{4-[4-(1,3-Dioxo-1,3-dihydro-i...)
Affinity DataKi:  213nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor of rat hippocampus using [3H]-8-hydroxy-2-(di-n-propylamine) tetralin (8-OH-DPAT) as a radio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50007171(CHEMBL316090 | N-(4-{4-[4-(1,3-Dioxo-1,3-dihydro-i...)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity towards alpha-1 adrenergic receptor of rat frontal cortex using [3H]- WB- 4101 as a radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed