Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 16 hits in this display
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
BDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50154009(Acetic acid 17-acetyl-6-chloro-10,13-dimethyl-3-ox...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
IC50: 259nMAssay Description:Antagonist activity at human AR AF2 assessed as inhibition of fluorescent-labelled D11-FxxLF peptide Co-activator to receptor by TR-FRET assayMore data for this Ligand-Target Pair
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
IC50: 631nMAssay Description:Inhibitory concentration against recombinant rat androgen receptor expressed in Escherichia coli using [3H]methyltrienolone (R 1881)More data for this Ligand-Target Pair
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)
BDBM50094569(6-chloro-3,20-dioxo-1beta,2beta-dihydro-3'H-cyclop...)